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C 101248
CAS No. 361368-24-3
C 101248( —— )
Catalog No. M37356 CAS No. 361368-24-3
C 101248 is a selective and potent inhibitor targeting both mouse and human tandem pore domain halothane-inhibited K+ channel 1 (THIK-1, IC50= 50 nM), without affecting the K2P family members (TREK-1, TWIK-2) and Kv2.1.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 10MG | 331 | Get Quote |
|
| 50MG | 1343 | Get Quote |
|
| 500MG | Get Quote | Get Quote |
|
| 1G | Get Quote | Get Quote |
|
Biological Information
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Product NameC 101248
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NoteResearch use only, not for human use.
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Brief DescriptionC 101248 is a selective and potent inhibitor targeting both mouse and human tandem pore domain halothane-inhibited K+ channel 1 (THIK-1, IC50= 50 nM), without affecting the K2P family members (TREK-1, TWIK-2) and Kv2.1.
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DescriptionKCNK13-IN-1 (example 71), a KCNK13 antagonist, is an anti-inflammatory agent, with an IC50 of <200 nM for IL-1 β.
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In Vitro——
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In Vivo——
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Synonyms——
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PathwayOthers
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TargetOther Targets
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RecptorOthers
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Research Area——
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Indication——
Chemical Information
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CAS Number361368-24-3
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Formula Weight292.3
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Molecular FormulaC15H12N6O
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Purity>98% (HPLC)
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Solubility——
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SMILESNC1=NON=C1C2=NC3=CC=CC=C3N2CC4=CC=NC=C4
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1. Roland BüRLI, et al. Novel compounds. Patent WO2022167819.
molnova catalog
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